Resumen de investigación: GLP-2 is an imbalanced dual GIP/Agonista del receptor GLP-1 exhibiting biased agonism with reduced β-arrestin recruitment at GLP-1R. CAS 2023788-19-2. 39-amino acid peptide with C20 fatty diacid for ~5-day half-life. Published in JCI Insight and PNAS. Péptido solo para investigación.
GLP-2
Dual GIP/Agonista del receptor GLP-1 — Solo para investigación
GLP-2 is a 39-amino acid synthetic dual GIP/Agonista del receptor GLP-1 classified as an imbalanced twincretin peptide. CAS Registry Number: 2023788-19-2. Molecular weight: ~4,813.45 Da. Molecular formula: C₂₂₅H₃₄₈N₄₈O₆₈. Compuesto para investigación supplied as lyophilized powder solo para uso de investigación.
Detalles del producto
- Compuesto: GLP-2
- Clasificación: Dual incretin receptor agonist
- Pureza: >99% (HPLC verified)
- Forma: Polvo liofilizado
- Pruebas: Ver COA (Verificado por Janoshik) →
Estudios de investigación
(solo con fines educativos)
Imbalanced dual GIP/Agonista del receptor GLP-1 profile
Willard FS, Douros JD, Gabe MBN, et al. · JCI Insight
Investigated GLP-2’s pharmacological profile as a dual receptor agonist, examining binding affinity and signaling patterns at GIP and GLP-1 receptors.
Additional receptor signaling characterization
Min Q, Bhatt DK, Mercer AJ, et al. · PNAS
Characterized signaling profiles using receptor-response assays, including cAMP readouts and receptor internalization measurements.
📚 Ver investigación publicada sobre GLP-2 →
Citas revisadas por pares de PubMed, solo con fines educativos
FOR RESEARCH USE ONLY
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